发明名称 CYCLIZATION PROCESS
摘要 PROBLEM TO BE SOLVED: To provide a method of very high volume efficiency for producing a racemate, azetidine-2-carboxylic acid. SOLUTION: A cyclization process from 4-amino-2-halobutyric acid to azetidine-2-carboxylic acid by which 20 g or more of the 4-amino-2-halobutyric acid are cyclized per 1 liter of the reaction mixture is provided. COPYRIGHT: (C)2009,JPO&INPIT
申请公布号 JP2009062392(A) 申请公布日期 2009.03.26
申请号 JP20080290610 申请日期 2008.11.13
申请人 ASTRAZENECA AB 发明人 PARRATT JULIAN SIMON;TAYLOR STEPHEN JOHN CLIFFORD
分类号 C07D205/04;A01D46/20;A01D46/24;B66F11/04;C07D205/08;G05D16/02 主分类号 C07D205/04
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