发明名称 |
6-SUBSTITUTED NICOTINAMIDE DERIVATIVES AS OPIOID RECEPTOR ANTAGONISTS |
摘要 |
A compound of the formula (I) or a pharmaceutically acceptable salt, enantiomer, racemate, diastereomers or mixtures thereof, or a solvate thereof, formulations and methods of use thereof, as opioid receptor antagonists are disclosed wherein the variables are as described herein.
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申请公布号 |
US2009023785(A1) |
申请公布日期 |
2009.01.22 |
申请号 |
US20080169057 |
申请日期 |
2008.07.08 |
申请人 |
PEDREGAL-TERCERO CONCEPCION;SIEGEL MILES GOODMAN;STUCKY RUSSELL DEAN;TAKEUCHI KUMIKO |
发明人 |
PEDREGAL-TERCERO CONCEPCION;SIEGEL MILES GOODMAN;STUCKY RUSSELL DEAN;TAKEUCHI KUMIKO |
分类号 |
A61K31/44;A61K31/166;A61K31/4427;A61P1/08;A61P3/04;A61P15/00;A61P17/04;A61P25/24;A61P25/30;C07D213/82;C07D401/12;C07D405/12;C07D409/12 |
主分类号 |
A61K31/44 |
代理机构 |
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代理人 |
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地址 |
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