发明名称 QUINAZOLIN-OXIME DERIVATIVES AS HSP90 INHIBITORS
摘要 Compounds of general formula (I); or a stereoisomers, tautomers, pharmaceutically acceptable salts, or prodrugs thereof, wherein R1, R2, R3, R4, R5, R6, R8 and R9 are as defined herein, are useful for the treatment of diseases and conditions which are mediated by excessive or inappropriate Hsp90 activity such as cancers, viral infection and inflammatory diseases or conditions.
申请公布号 WO2008142720(A2) 申请公布日期 2008.11.27
申请号 WO2008IT00326 申请日期 2008.05.15
申请人 DAC SRL;COURTNEY, STEPHEN MARTIN;WHITTAKER, MARK;MATHER, OWEN CLIFFORD;YARNOLD, CHRISTOPHER JOHN;BARKER, OLIVER ROBIN;MONTALBETTI, CHRISTIAN ALDO GEORGES NAPOLEON;HESTERKAMP, THOMAS;GARDINER, MIHALY DANIEL 发明人 COURTNEY, STEPHEN MARTIN;WHITTAKER, MARK;MATHER, OWEN CLIFFORD;YARNOLD, CHRISTOPHER JOHN;BARKER, OLIVER ROBIN;MONTALBETTI, CHRISTIAN ALDO GEORGES NAPOLEON;HESTERKAMP, THOMAS;GARDINER, MIHALY DANIEL
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