发明名称 HETEROCYCLYL-SUBSTITUTED ANTI-HYPERCHOLESTEROLEMIC COMPOUNDS
摘要 This invention provides cholesterol absorption inhibitors of Formula I: and the pharmaceutically acceptable salts thereof, wherein R<SUP>12</SUP> is a hydroxylated alkyl group and R<SUP>9</SUP> contains a heterocyclic ring. The compounds are useful for lowering plasma cholesterol levels, particularly LDL cholesterol, and for treating atherosclerosis and preventing atherosclerotic disease events.
申请公布号 WO2008057336(A3) 申请公布日期 2008.09.18
申请号 WO2007US22895 申请日期 2007.10.30
申请人 MERCK & CO., INC.;MORRIELLO, GREGORI, J.;DEVITA, ROBERT, J.;MOYES, CHRISTOPHER, R. 发明人 MORRIELLO, GREGORI, J.;DEVITA, ROBERT, J.;MOYES, CHRISTOPHER, R.
分类号 A01N43/00;A61K31/397 主分类号 A01N43/00
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