Process for the preparation of ezetimibe and derivatives thereof
摘要
The present invention relates to the method of preparing of ezetimibe and in particular to novel intermediates for its synthesis and an improved process for preparing such intermediates. Said intermediates may be obtained in high yields and purity in a fast and cost efficient manner. The present invention relates to a novel crystalline form of ezetimibe as well.
申请公布号
EP1953140(A1)
申请公布日期
2008.08.06
申请号
EP20070001537
申请日期
2007.01.24
申请人
KRKA
发明人
STIMAC, ANTON;MOHAR, BARBARA;STEPHAN, MICHEL;BEVC, MOJCA;ZUPET, ROK;GARTNER, ANDREJ;KROSELJ, VESNA;SMRKOLJ, MATEJ