发明名称 Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
摘要 The invention relates to the use of 4-aminopyrimidines of formula (I), in which R<SUP>1</SUP>-H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkinyl, R<SUP>2</SUP>-H, halogen, cyano, alkyl, alkylhalide, alkenyl, alkinyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, whereby the hydrocarbon chain in R<SUP>1 </SUP>and/or R<SUP>2 </SUP>can be substituted as given in the description, R<SUP>1 </SUP>and R<SUP>2 </SUP>can form, together with the carbon atom to which they are bonded, a 5-7-membered ring which can contain one to three same or different heteroatoms selected from the group O, N or S, R<SUP>3</SUP>-H, halogen, cyano, hydroxy, mercapto, azido, alkyl, alkenyl, alkinyl, alkylhalide, -O-D, -S(O)<SUB>m</SUB>-D, ON-CR<SUP>a</SUP>R<SUP>b</SUP>, CR<SUP>c</SUP>-NOR<SUP>a</SUP>, NR<SUP>c</SUP>N-CR<SUP>a</SUP>R<SUP>b</SUP>, NR<SUP>a</SUP>R<SUP>b</SUP>, NR<SUP>c</SUP>NR<SUP>a</SUP>R<SUP>b</SUP>, NOR<SUP>a</SUP>, NR<SUP>c</SUP>C(-NR<SUP>c</SUP>)NR<SUP>a</SUP>R<SUP>b</SUP>, NR<SUP>c</SUP>C(-O)NR<SUP>a</SUP>R<SUP>b</SUP>, NR<SUP>a</SUP>CN, -NR<SUP>a</SUP>C(-O)R<SUP>c</SUP>, NR<SUP>a</SUP>C(-NOR<SUP>c</SUP>)R<SUP>c'</SUP>, OC(-O)R<SUP>a</SUP>, C(-NOR<SUP>c</SUP>)NR<SUP>a</SUP>R<SUP>b</SUP>, CR<SUP>c</SUP>(-NNR<SUP>a</SUP>R<SUP>b</SUP>), C(-O)NR<SUP>a</SUP>R<SUP>b</SUP>, C(-O)R<SUP>a</SUP>, CO<SUB>2</SUB>R<SUP>a</SUP>, C(-O)NR<SUP>z</SUP>R<SUP>b</SUP>, C(-O)-N-OR<SUP>b</SUP>, C(-S)-NR<SUP>z</SUP>R<SUP>b</SUP>, C(-O)NR<SUP>a</SUP>-NR<SUP>z</SUP>R<SUP>b</SUP>, C(-N-NR<SUP>z</SUP>R<SUP>c</SUP>)NR<SUP>a</SUP>R<SUP>b</SUP>, C(-NOR<SUP>b</SUP>)R<SUP>a</SUP>, C(-N-NR<SUP>z</SUP>R<SUP>b</SUP>)R<SUP>a</SUP>, CR<SUP>a</SUP>R<SUP>b</SUP>-OR<SUP>z</SUP>, CR<SUP>a</SUP>R<SUP>b</SUP>-NR<SUP>z</SUP>R<SUP>c</SUP>, ON(-CR<SUP>a</SUP>R<SUP>b</SUP>), NR<SUP>a</SUP>(C(-O)R<SUP>b</SUP>), NR<SUP>a</SUP>(C(-O)OR<SUP>b</SUP>), C(-NR<SUP>a</SUP>)NR<SUP>z</SUP>R<SUP>b</SUP>, C(-0)-NR<SUP>z</SUP>R<SUP>b</SUP>) NR<SUP>a</SUP>(C(-O)-NR<SUP>z</SUP>R<SUP>b</SUP>), NR<SUP>a</SUP>(C(-NR<SUP>c</SUP>)R<SUP>b</SUP>), NR<SUP>a</SUP>(N-CR<SUP>c</SUP>R<SUP>b</SUP>), NR<SUP>a</SUP>-NR<SUP>z</SUP>R<SUP>b</SUP>, -NR<SUP>z</SUP>-OR<SUP>a</SUP>, NR<SUP>a</SUP>(C(-NR<SUP>c</SUP>)-NR<SUP>z</SUP>R<SUP>b</SUP>), NR<SUP>a</SUP>(C(-NOR<SUP>c</SUP>)R<SUP>b</SUP>) D=alkyl, alkenyl, alkinyl, alkylhalide, cycloalkyl, five- or six-membered saturated, partly-unsaturated or aromatic mono- or bicyclic heterocycles, containing one to four heteroatoms from the group O, N or S, one of the groups G1 or G2, whereby m, x, R<SUP>a</SUP>, R<SUP>b</SUP>, R<SUP>c</SUP>, R<SUP>d</SUP>, R<SUP>e</SUP>, R<SUP>z</SUP>, Y, Z are as defined in the description and the aliphatic, alicyclic or aromatic groups R<SUP>3</SUP>, R<SUP>a</SUP>, R<SUP>b</SUP>, R<SUP>c</SUP>, R<SUP>d </SUP>or R<SUP>e </SUP>can be substituted as given in the description for the prevention of fungal pests, novel 4-aminopyridines, method for production of said compounds and agents comprising the same.
申请公布号 US2008176744(A1) 申请公布日期 2008.07.24
申请号 US20060885822 申请日期 2006.03.08
申请人 BASF AKTIENGESELLSCHAFT 发明人 SCHWOGLER ANJA;RHEINHEIMER JOACHIM;GRAMMENOS WASSILIOS;GROTE THOMAS;HUNGER UDO;MULLER BERND;SCHAFER PETER;SCHIEWECK FRANK
分类号 A01N43/54;A01C1/06;C07D239/42 主分类号 A01N43/54
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