发明名称 DIRECT AMINOLYSIS
摘要 In some aspects, the present invention provides a method of preparing a compound of the formula (I) comprising reacting a mesylate compound of the formula (II) by direct aminolysis with a reagent comprising ammonia. The reaction is preferably carried out in a solvent, such as an alcohol, and is preferably carried out in a sealed vessel such as a Parr reactor or the like.
申请公布号 KR20080031489(A) 申请公布日期 2008.04.08
申请号 KR20087004939 申请日期 2008.02.28
申请人 PFIZER PRODUCTS INC. 发明人 LI ZHENGONG BRYAN
分类号 C07C209/22;C07C211/36;C07D205/04 主分类号 C07C209/22
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