| 发明名称 |
Novel method for synthesising derivatives of (2S, 3AS, 7AS)-1-[(S)-alanyl]-octahydro,-1H-indole-2-carboxylic acid and the use thereof for perindopril synthesis |
| 摘要 |
<p>Disclosed is a method for synthesising compounds of formula (I), wherein R1 is a hydrogen atom or a linear or branched (c1-C6) alkyl or benzyl group and R2 is an amine function protecting group. The use of said compounds for synthesising perindopril and the pharmaceutically acceptable salts thereof are also disclosed.</p> |
| 申请公布号 |
NZ541423(A) |
申请公布日期 |
2008.03.28 |
| 申请号 |
NZ20040541423 |
申请日期 |
2004.02.27 |
| 申请人 |
LES LABORATOIRES SERVIER |
发明人 |
DUBUFFET, THIERRY;LANGLOIS, PASCAL |
| 分类号 |
C07D209/42;C07K5/02;C07K5/06;(IPC1-7):C07D209/42 |
主分类号 |
C07D209/42 |
| 代理机构 |
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