发明名称 |
PYRIDAZINONE DERIVATIVE AND PDE INHIBITOR COMPRISING THE SAME AS ACTIVE INGREDIENT |
摘要 |
PROBLEM TO BE SOLVED: To provide a novel pyridazinone derivative useful as a pharmaceutical product having a phosphodiesterase inhibitory activity. SOLUTION: A phosphodiesterase (PDE) inhibitor contains the pyridazinone derivative represented by formula (1) [wherein Heterocycle represents a benzoxazole ring or a benzothiazole ring], an optical isomer thereof, a pharmacologically acceptable salt thereof or a hydrate thereof as an active ingredient. COPYRIGHT: (C)2008,JPO&INPIT
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申请公布号 |
JP2008063265(A) |
申请公布日期 |
2008.03.21 |
申请号 |
JP20060241618 |
申请日期 |
2006.09.06 |
申请人 |
KYORIN PHARMACEUT CO LTD |
发明人 |
KONO YASUSHI;ADAMS DAVID R |
分类号 |
C07D403/04;A61K31/501;A61P1/04;A61P3/04;A61P3/06;A61P3/10;A61P7/02;A61P9/04;A61P9/10;A61P9/12;A61P11/00;A61P11/02;A61P11/06;A61P15/10;A61P17/02;A61P19/02;A61P25/00;A61P25/14;A61P25/16;A61P25/18;A61P25/24;A61P25/28;A61P29/00;A61P37/08;A61P43/00;C07D413/04;C07D417/04 |
主分类号 |
C07D403/04 |
代理机构 |
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