发明名称 COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF
摘要 The present invention provides novel beta-secretase inhibitors of the general formula (I), where the variables A1, A2, L 1, L2, L3, R1, R2, R3, R4, R5, R6 and R7 are as defined in the claims, a method for their use in treating Alzheimer's disease, and methods for their use in reducing memapsin 2 catalytic activity.
申请公布号 KR20080015079(A) 申请公布日期 2008.02.18
申请号 KR20077025947 申请日期 2007.11.08
申请人 COMENTIS, INC.;OKLAHOMA MEDICAL RESEARCH FOUNDATION;PURDUE RESEARCH FOUNDATION;THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 发明人 GHOSH ARUN K.;KUMARAGURUBARAN NAGASWAMY;LIU CHUNFENG;DEVASAMUDRAM THIPPESWAMY;LEI HUI;SWANSON LISA;ANKALA SUDHA;TANG JORDAN;BILCER GEOFFREY
分类号 C07C233/78;C07C237/24;C07C311/08;C07C311/29 主分类号 C07C233/78
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