发明名称 CRYSTALLINE FORM OF A QUINOLINONE-CARBOXAMIDE COMPOUND
摘要 The invention provides a crystalline hydrochloride salt of 1-isopropyl-2-oxo-1,2-dihydroquinoline-3-carboxylic acid {(1S,3R,5R)-8-[(R)-2-hydroxy-3-(methanesulfonyl-methyl-amino)propyl]-8-azabicyclo[3.2.1]oct-3-yl}amide or a solvate thereof. The invention also provides pharmaceutical compositions comprising such crystalline salt forms, methods of using such crystalline salt forms to treat diseases associated with 5-HT4 receptor activity, and processes useful for preparing such crystalline salt forms.
申请公布号 EP1874766(A2) 申请公布日期 2008.01.09
申请号 EP20060740692 申请日期 2006.04.05
申请人 THERAVANCE, INC. 发明人 FATHEREE, PAUL R.;TURNER, S. DEREK;GOLDBLUM, ADAM;CHAO, ROBERT;GENOV, DANIEL
分类号 C07D451/04;A61K31/40;A61P1/00 主分类号 C07D451/04
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