发明名称 |
PRODRUG ERß-SELECTIVE SUBSTANCES, METHODS FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID COMPOUNDS |
摘要 |
The invention relates to a prodrugs of 9a-substituted estratrienes of general formula (I), wherein the Z group is linked to a steroid, (I). The invention also relates to a methods for the production thereof, pharmaceutical compositions which contain said compounds, and to the use thereof. Said inventive compounds of general formula (I) do not bond with the oestrogen receptor alpha and/ or beta but they bond with carboanhydrases and inhibitors of said enzymes. |
申请公布号 |
WO2007062877(A3) |
申请公布日期 |
2007.11.08 |
申请号 |
WO2006EP11729 |
申请日期 |
2006.11.27 |
申请人 |
BAYER SCHERING PHARMA AKTIENGESELLSCHAFT;MUELLER, GERD;KOSEMUND, DIRK;WYRWA, RALF |
发明人 |
MUELLER, GERD;KOSEMUND, DIRK;WYRWA, RALF |
分类号 |
C07J41/00;A61K31/565;A61P5/28;A61P5/32;A61P15/00;A61P19/10 |
主分类号 |
C07J41/00 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|