发明名称 AN IMPROVED PROCESS FOR THE PREPARATION OF OXCARBAZEPINE AND RELATED INTERMEDIATES
摘要 A process for preparing Oxcarbazepine III comprising: a) reacting oximinostilbene IV with chlorosulfonyl isocyanate in an inert organic solvent and isolating compound V b) hydrolyzing compound V to form crude Oxcarbazepine III c) purifying oxcarbazepine.
申请公布号 WO2005122671(A3) 申请公布日期 2007.11.08
申请号 WO2005CA00932 申请日期 2005.06.16
申请人 APOTEX PHARMACHEM INC.;CHE, DAQING;CORELLI-RENNIE, NADIA;GUNTOORI, BHASKAR, REDDY;FAUGHT, JODY 发明人 CHE, DAQING;CORELLI-RENNIE, NADIA;GUNTOORI, BHASKAR, REDDY;FAUGHT, JODY
分类号 C07D223/22;A61K31/55;C07D223/18;C07D223/26;C07D223/28;C07D223/30 主分类号 C07D223/22
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