发明名称 |
Subcutaneous delivery system, process for the preparation of the same and use of the same for the treatment of cholinergic deficient disorders |
摘要 |
The present invention relates to a subcutaneous delivery system comprising a biodegradable polymeric matrix and at least one of the pharmacologically active substances of general formula (I): wherein A represents an amino group -NH<SUB>2 </SUB>or an ammonium group -NH<SUB>3</SUB>+ or a residue of general formula (II): wherein each of X<SUB>1 </SUB>to X<SUB>5 </SUB>represents, independently, an hydrogen atom, a linear or branched C<SUB>1 </SUB>to C<SUB>6 </SUB>alkyl group, a linear or branched C<SUB>1 </SUB>to C<SUB>6 </SUB>alkyloxy group, a hydroxyl group -OH, an amino group -NH<SUB>2</SUB>, a primary or secondary C<SUB>1 </SUB>to C<SUB>6 </SUB>alkylamino group, a halogen atom, a nitro group -NO<SUB>2</SUB>; said substance being embedded into said matrix. It relates also to a process for its preparation and to its use for the preparation of a medicament.
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申请公布号 |
US2007059369(A1) |
申请公布日期 |
2007.03.15 |
申请号 |
US20040549167 |
申请日期 |
2004.03.15 |
申请人 |
MAUVERNAY ROLLAND-YVES;PORCHET HERVE;SCALFARO PIETRO;HEIMGARTNER FREDERIC;DUCREY BERTRAND;PFEFFERLE FRANCOIS;CAPANCIONI SERGIO;MC CORMICK MARK |
发明人 |
MAUVERNAY ROLLAND-YVES;PORCHET HERVE;SCALFARO PIETRO;HEIMGARTNER FREDERIC;DUCREY BERTRAND;PFEFFERLE FRANCOIS;CAPANCIONI SERGIO;MC CORMICK MARK |
分类号 |
A61K31/473;A61K;A61K9/00;A61K9/14;A61K9/20;A61K31/465;A61P21/00;A61P25/28;A61P39/00 |
主分类号 |
A61K31/473 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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