发明名称 PROCESS FOR THE PREPARATION OF N-[(1-NBUTYL-4-PIPERIDYL)METHYL] -3,4-DIHYDRO -2H-[1,3] OXAZINO[3,2-A] INDOLE-10-CARBOXAMIDE AND SALTS AND INTERMEDIATES IN THE PROCESS
摘要 <p>A process for the preparation of SB 207266 or a pharmaceutically acceptable salt thereof, which process comprises the reaction of N-(1-n butyl-4- piperidyl)methylamine with a compound of formula (A), wherein R is alkyl.</p>
申请公布号 CA2263480(C) 申请公布日期 2007.03.06
申请号 CA19972263480 申请日期 1997.08.11
申请人 SMITHKLINE BEECHAM P.L.C. 发明人 GUEST, DAVID WILLIAM;STRACHAN, JOHN BRYCE;FEDOULOFF, MICHAEL;SMITH, GILLIAN ELIZABETH
分类号 C07D498/04;C07D209/42 主分类号 C07D498/04
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