发明名称 PARTIAL OR FULL A1 AGONISTS - N6 HETEROCYCLIC 5'-THIO SUBSTITUTED ADENOSINE DERIVATIVES
摘要 N6 heterocyclic 5' modified adenosine derivatives that are adenosine A1 receptor partial or full agonists, and as such, are useful for modifying cardiac activity, modifying adipocyte functio n, treating central nervous system disorders, and treating diabetic disorders and obesity in mammals, and especially in humans.
申请公布号 CA2389264(C) 申请公布日期 2007.03.06
申请号 CA20002389264 申请日期 2000.12.01
申请人 CV THERAPEUTICS, INC. 发明人 PALLE, VENKATA P.;ZABLOCKI, JEFF A.;VARKHEDKAR, VAIBHAV;BELARDINELLI, LUIZ;IBRAHIM, PRABHA
分类号 C07H19/16;C07H19/167;A61K9/08;A61K9/20;A61K31/7076;A61P3/04;A61P3/10;A61P9/00;A61P9/04;A61P9/10;A61P25/00;A61P25/08;A61P43/00 主分类号 C07H19/16
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