发明名称 PLEUROMUTILIN DERIVATIVES USEFUL AS ANTIBACTERIALS
摘要 <p>The present invention relates to compounds selected from the group consisting of 14-0- [((Mono- or dialkylamino)-cycloalkylsulfanyl- or -cycloalkyl-oxy)-acetyl, -thioacetyl or - imino-oxy]-mutilins, 14-O-[((Cycloalkyl- or heterocyclylamino)-cycloalkylsulfanyl- or - cycloalkyl-oxy)-acetyl, -thioaceyl or -imino-oxy]-mutilins, 14-O-[((Heterocyc-N-yl- cycloalkyl)-sulfanyl- or -oxy)-acetyl, -thioacetyl or -imino-oxy]-mutilins, 14-O-[(((Mono- or dialkylamino)-cycloalkyl)-alkylsulfanyl- or -alkyl-oxy)-acetyl, -thioacetyl or -imino-oxy]- mutilins, 14-O-[(((Cycloalkyl- or heterocyclylamino)-cycloalkyl)-alkylsulfanyl- or -alkyl- oxy)-acetyl, -thioacetyl or -imino-oxy]-mutilins, and 14-O-[((Heterocyc-N-yl-cycloalkyl)- alkylsulfanyl- or -alkyl-oxy)-acetyl, -thioacetyl or -imino-oxy]-mutilins, and their use as pharmaceuticals.</p>
申请公布号 WO2007014409(A1) 申请公布日期 2007.02.08
申请号 WO2006AT00318 申请日期 2006.07.26
申请人 NABRIVA THERAPEUTICS FORSCHUNGS GMBH;MANG, ROSEMARIE;BERNER, HEINZ 发明人 MANG, ROSEMARIE;BERNER, HEINZ
分类号 C07C323/52;A61K31/10;A61P31/04 主分类号 C07C323/52
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