发明名称 PYRROLOPYRIMIDINONE DERIVATIVE
摘要 A compound represented by the following formula, which has inhibitory activity against GSK-3. (I) In the formula, A1 and A3 each is a single bond or an aliphatic hydrocarbon; A2 and A4 each is a single bond, CO, COO, etc.; G1 is a single bond, alicyclic hydrocarbon, aromatic hydrocarbon, etc.; G2 is hydrogen, an aliphatic hydrocarbon, alicyclic hydrocarbon, aromatic hydrocarbon, etc.; A5 is a single bond or NR; R2 is hydrogen, halogeno, an aliphatic hydrocarbon, etc.; A6 is a single bond, NR, CO, etc.; and R3 is hydrogen, halogeno, nitro, a saturated aliphatic hydrocarbon, etc.; provided that R is hydrogen or a lower aliphatic hydrocarbon group.
申请公布号 KR20060118416(A) 申请公布日期 2006.11.23
申请号 KR20067003712 申请日期 2006.02.23
申请人 TEIJIN PHARMA LIMITED 发明人 TSUTSUMI TAKAHARU;SUGIURA SATOSHI;KOGA MASAHIRO;MATSUMOTO YOSHIYUKI;ISHII TOSHIHIRO;NAKANO AKIRA;UNOKI GEN;SAKAI YURI;TAKARADA REIKO;OGAWA HIROKO
分类号 C07D487/04;A61K31/519;A61P3/10;A61P17/14;A61P25/24;A61P25/28;A61P29/00;A61P35/00;A61P37/02;A61P43/00;C07D487/02 主分类号 C07D487/04
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