发明名称 PROCESSES FOR THE PREPARATION OF ROCURONIUM BROMIDE AND INTERMEDIATES THEREOF
摘要 A novel process for preparing (2beta,3alpha,5alpha,16alpha,17beta)-17-acetoxy-3-hydroxy-2-(4-morpholinyl)-16-(1-pyrrolidinyl) androstane, a known intermediate in the synthesis of the skeletal muscle relaxant rocuronium bromide, is disclosed.
申请公布号 WO2005068487(A3) 申请公布日期 2006.02.02
申请号 WO2005IL00049 申请日期 2005.01.13
申请人 CHEMAGIS LTD.;ADAR, ELIEZER;SONDACK, DAVID;FRIEDMAN, ODED;MANASCU, IOSEF;FIZITZKI, TAMIR;FREGER, BORIS;ARAD, ODED;WEISMAN, ALEXANDER;KASPI, JOSEPH 发明人 ADAR, ELIEZER;SONDACK, DAVID;FRIEDMAN, ODED;MANASCU, IOSEF;FIZITZKI, TAMIR;FREGER, BORIS;ARAD, ODED;WEISMAN, ALEXANDER;KASPI, JOSEPH
分类号 C07J11/00;A61K31/58;C07J43/00 主分类号 C07J11/00
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