发明名称 |
ЛЕКАРСТВЕННОЕ СРЕДСТВО ПРОТИВ ГИПЕРАКТИВНОГО МОЧЕВОГО ПУЗЫРЯ, ВКЛЮЧАЮЩЕЕ ПРОИЗВОДНОЕ АНИЛИДА УКСУСНОЙ КИСЛОТЫ В КАЧЕСТВЕ АКТИВНОГО ИНГРЕДИЕНТА |
摘要 |
(R)-2-(2-aminothiazol-4-yl)-4'-Ä2-Ä(2-hydroxy-2-phenylethyl)aminoÜethylÜacetic acid anilide or its salt shows a potent bladder relaxation effect in "isolated rat bladder smooth muscle relaxation test", dose-dependently lowers the contraction frequency of rhythmic bladder contractions in "rat rhythmic bladder contraction measurement test" and, moreover, prolongs the urination intervals in "urination functions measurement test on cyclophosphamide-induced overactive bladder model rat". Owing to these effects, the above compound is useful as a remedy for ovaractive bladder. |
申请公布号 |
RU2005117367(A) |
申请公布日期 |
2006.01.20 |
申请号 |
RU20050117367 |
申请日期 |
2003.11.04 |
申请人 |
АСТЕЛЛАС ФАРМА ИНК. (JP) |
发明人 |
ТАКАСУ Тосиюки (JP);САТО Суити (JP);УКАЙ Масаси (JP);МАРУЯМА Тацу (JP) |
分类号 |
A61K31/426;A61P13/00;A61P13/10;C07D277/40 |
主分类号 |
A61K31/426 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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