发明名称 |
6-SUBSTITUTED PYRIDOINDOLONE DERIVATIVES PRODUCTION AND THERAPEUTIC USE THEREOF |
摘要 |
<p>The invention relates to compounds of formula (I), where R1 = H, C1-C4 alkyl, -(CH2)mOH, -(CH2)mCN, or -(CH2)mNR9R10, R2 =H, or C1-C4 alkyl, R3 = phenyl substituted by R6, R7, or R8, R4 = a group of formula (a), a heterocyclic group selected from formulae (b), (c), or (d) and R5 = H, or C1-C4 alkyl. The invention further relates to a production method and therapeutic application thereof.</p> |
申请公布号 |
WO2005108398(A1) |
申请公布日期 |
2005.11.17 |
申请号 |
WO2005FR00971 |
申请日期 |
2005.04.20 |
申请人 |
SANOFI-AVENTIS;BOURRIE, BERNARD;CASELLAS, PIERRE;CIAPETTI, PAOLA;DEROCQ, JEAN MARIE;JEGHAM, SAMIR;MUNEAUX, YVETTE;WERMUTH, CAMILLE-GEORGE |
发明人 |
BOURRIE, BERNARD;CASELLAS, PIERRE;CIAPETTI, PAOLA;DEROCQ, JEAN MARIE;JEGHAM, SAMIR;MUNEAUX, YVETTE;WERMUTH, CAMILLE-GEORGE |
分类号 |
A61P35/00;A61K31/407;A61K31/437;A61K31/4412;C07D471/04;(IPC1-7):C07D471/04 |
主分类号 |
A61P35/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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