发明名称 PROCESS FOR THE PREPARATION OF TELMISARTAN
摘要 <p>An improved process for the preparation of telmisartan, or a pharmaceutically acceptable salt thereof, comprises subjecting 1H-Benzimidazole-2-n-propyl-4-methyl-6-(1'-methyl benimidazole-2'yl) of formula (II) and methyl-4-(bromomethyl) biphenyl-2-carboxylate of formula (III) to condensation and hydrolysis in a single step.</p>
申请公布号 WO2005108375(A1) 申请公布日期 2005.11.17
申请号 WO2005GB01799 申请日期 2005.05.10
申请人 CIPLA LIMITED;KANKAN, RAJENDRA, NARAYANRAO;RAO, DHARMARAJ, RAMACHANDRA;SRINIVAS, PATHI, L.;RAVIKUMAR, PUPPALA;TURNER, CRAIG, ROBERT 发明人 KANKAN, RAJENDRA, NARAYANRAO;RAO, DHARMARAJ, RAMACHANDRA;SRINIVAS, PATHI, L.;RAVIKUMAR, PUPPALA
分类号 A61K31/4184;C07D235/18;C07D235/20;(IPC1-7):C07D235/18;A61P9/04;A61K31/418;A61P9/02 主分类号 A61K31/4184
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