发明名称 |
Substituted arylamine derivatives and methods of use |
摘要 |
Selected compounds are effective for prophylaxis and treatment of diseases, such as angiogenesis mediated diseases. The invention encompasses novel compounds, analogs, prodrugs and pharmaceutically acceptable derivatives thereof, pharmaceutical compositions and methods for prophylaxis and treatment of diseases and other maladies or conditions involving, cancer and the like. The subject invention also relates to processes for making such compounds as well as to intermediates useful in such processes.
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申请公布号 |
US2005153960(A1) |
申请公布日期 |
2005.07.14 |
申请号 |
US20040996035 |
申请日期 |
2004.11.22 |
申请人 |
AMGEN INC. |
发明人 |
ELBAUM DANIEL;ASKEW BENNY C.JR.;BOOKER SHON;GERMAIN JULIE;HABGOOD GREGORY J.;HANDLEY MICHAEL;KIM TAE-SEONG;LI AIWEN;NISHIMURA NOBUKO;PATEL VINOD F.;YUAN CHESTER C.;KIM JOSEPH L.;CAI GUOLIN;CHEN GUOQING;CROGHAN MICHAEL;DI PIETRO LUCIAN V.;DOMINGUEZ CELIA;HUANG QI;SMITH LEON M.II;TASKER ANDREW;XI NING;XU SHIMIN |
分类号 |
A61K31/44;A61K31/4427;A61K31/443;A61K31/4436;A61K31/4439;A61K31/444;A61K31/4709;A61K31/4725;A61K31/496;A61K31/498;A61K31/501;A61K31/506;A61K31/517;A61K31/5377;A61K31/538;A61P1/04;A61P3/00;A61P3/04;A61P3/10;A61P9/00;A61P9/10;A61P11/00;A61P11/06;A61P15/00;A61P15/08;A61P17/00;A61P17/02;A61P17/06;A61P19/00;A61P19/02;A61P21/00;A61P25/28;A61P27/02;A61P27/06;A61P29/00;A61P31/12;A61P31/18;A61P31/22;A61P35/00;A61P35/02;A61P35/04;A61P37/02;A61P37/04;A61P37/08;A61P43/00;C07D213/81;C07D213/82;C07D237/04;C07D237/24;C07D401/12;C07D401/14;C07D405/12;C07D409/12;C07D413/12;C07D413/14;C07D417/12;C07D471/04;(IPC1-7):A61K31/538;A61K31/470;A61K31/454;C07D413/02;C07D41/02 |
主分类号 |
A61K31/44 |
代理机构 |
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