发明名称 PYRIDYL DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS
摘要 Methods of treating an SCD-mediated disease or condition in a mammal, preferably a human, are disclosed, wherein the methods comprise administering to a mammal in need thereof a compound of formula (I): wherein W, V, x, y, R<1>, R<2>, R<3>, R<4>, R<5>, R<6>, R<7>, R<7>a, R<8>, R<8>a, R<9>, R<9a>, R<10> and R<10a> are defined herein. Pharmaceutical compositions comprising the compounds of formula (I) are also disclosed.
申请公布号 WO2005011654(A2) 申请公布日期 2005.02.10
申请号 WO2004US24542 申请日期 2004.07.29
申请人 XENON PHARMACEUTICALS INC.;ABREO, MELWYN;HARVEY, DANIEL, F.;KONDRATENKO, MIKHAIL, A.,;LI, WENBAO;KAMBOJ, RAJENDER;KODUMURU, VISHNUMURTHY;WINTHER, MICHAEL, D.;GSCHWEND, HEINZ, W.;CHAKKA, NAGASREE;LIU, SHIFENG;SVIRIDOV, SERGUEI;SUN, SHAOYI 发明人 ABREO, MELWYN;HARVEY, DANIEL, F.;KONDRATENKO, MIKHAIL, A.,;LI, WENBAO;KAMBOJ, RAJENDER;KODUMURU, VISHNUMURTHY;WINTHER, MICHAEL, D.;GSCHWEND, HEINZ, W.;CHAKKA, NAGASREE;LIU, SHIFENG;SVIRIDOV, SERGUEI;SUN, SHAOYI
分类号 A61K31/00;A61K31/501;A61P3/06;C07D213/75;C07D213/76;C07D213/81 主分类号 A61K31/00
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