发明名称 PROCESS FOR PREPARATION OF PERINDOPRIL AND SALTS THEREOF
摘要 <p>A process for preparation of perindopril of formula (II) and salts thereof which is simple, safe, convenient and cost-effective. The process involves reaction of compound of formula (I), wherein X is chlorine or bromine with compound of formula (VII) wherein A signifies that the six-membered ring of the bicyclic system is either saturated or unsaturated, followed by catalytic hydrogenation to give the perindopril of formula (II).</p>
申请公布号 WO2004075889(A1) 申请公布日期 2004.09.10
申请号 WO2003IN00042 申请日期 2003.02.28
申请人 LUPIN LIMITED;DATTA, DEBASHISH;SINGH, GIRIJ, PAL;GODBOLE, HIMANSHU, MADHAV;SIYAN, RAJINDER, SINGH 发明人 DATTA, DEBASHISH;SINGH, GIRIJ, PAL;GODBOLE, HIMANSHU, MADHAV;SIYAN, RAJINDER, SINGH
分类号 C07C229/12;A61P9/12;C07C227/32;C07C227/34;C07D209/42;(IPC1-7):A61K31/404 主分类号 C07C229/12
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