发明名称 1,3-DIHYDRO-2H-INDOL-2-ONE DERIVATIVES AND THEIR USE AS LIGANDS FOR V1B OR V1B AND V1A ARGININE-VASOPRESSIN RECEPTORS
摘要 The invention relates to compounds of formula: as well as the possible salts thereof with mineral or organic acids, and the solvates and/or hydrates thereof, which have affinity for and selectivity towards the V1b receptors or towards both the V1b and V1a receptors of arginine-vasopressin. The invention also relates to the process for preparing them, to the intermediate compounds of formula (II) that are useful for preparing them, to pharmaceutical compositions containing them and to their use for the preparation of medicinal products.
申请公布号 EP1255751(B1) 申请公布日期 2004.06.16
申请号 EP20010907685 申请日期 2001.01.24
申请人 SANOFI-SYNTHELABO 发明人 ROUX, RICHARD;SERRADEIL-LE GAL, CLAUDINE;TONNERRE, BERNARD;WAGNON, JEAN
分类号 A61K;A61K31/404;A61K31/405;A61K31/496;A61K31/5377;A61P;A61P1/00;A61P1/18;A61P3/06;A61P3/08;A61P5/38;A61P5/50;A61P7/04;A61P9/00;A61P9/10;A61P9/12;A61P11/06;A61P13/02;A61P15/04;A61P15/12;A61P17/06;A61P25/00;A61P25/02;A61P25/06;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P27/12;A61P29/00;A61P35/00;A61P37/06;A61P37/08;A61P43/00;C07D;C07D207/12;C07D209/04;C07D209/34;C07D403/04;C07D403/14;C07D405/06;C07D405/14;(IPC1-7):C07D403/04 主分类号 A61K
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