发明名称 |
alpha-hydroxyarylbutanamine inhibitors of aspartyl protease |
摘要 |
Acylated alpha-hydroxyarylbutanamines and related sulfonamides, ureas and carbamates that inhibit aspartyl protease are disclosed, as are methods of treating diseases, particularly HIV, using these compounds. The compounds have the formula:A representative example is:
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申请公布号 |
US6696494(B2) |
申请公布日期 |
2004.02.24 |
申请号 |
US20010007235 |
申请日期 |
2001.10.22 |
申请人 |
ENANTA PHARMACEUTICALS, INC. |
发明人 |
OR YAT SUN;WANG GUOQIANG;ROUGAS JOHN;MATHEWS JUDE ELIZABETH;MULDOON KATE RYAN;BOYD VINCENT ALFRED;ECKSTEIN JENS WERNER;RIESINGER STEVEN WAYNE |
分类号 |
C07C235/42;C07C235/52;C07C235/74;C07C235/76;C07C235/84;C07C237/12;C07C237/36;C07C271/22;C07C275/24;C07C275/28;C07C275/30;C07C311/06;C07C311/19;C07C311/51;C07C323/60;C07C333/04;C07D213/65;C07D213/71;C07D215/36;C07D233/76;C07D261/08;C07D271/12;C07D279/30;C07D295/192;C07D295/215;C07D307/20;C07D311/24;C07D333/34;(IPC1-7):A61K31/165;C07C211/27 |
主分类号 |
C07C235/42 |
代理机构 |
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