| 摘要 |
The present invention is directed to an arylation of a nuclophile by reactin g the nucleophile with a substrate aromatic compound ArX in the presence of a copper catalyst, a base and water, wherein Ar is aryl, heteroaryl or alkenyl , X is halo, sulfonate or phosphonate, the base comprises an alkaline earth carbonate, bicarbonate, hydroxide or phosphate, and the copper catalyst comprises a copper atom or ion and a ligand.
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