发明名称 ANTIPARASITIC PYRAZOLS
摘要 <p>The compounds are used in the composition of antiparasitic formulations. They have the formula where R1 is 2,4,6-trisubstituted phenyl or 3,5-disubstituted pyridin-2-yl; R3 is C1-C4 alkyl, optionally substituted by hydroxy or by one or more halo, cyano, alkanoyl or phenyl; R5 is hydrogen, C1-C4 alkyl, amino or halo; R2 and R4 are independant from each other and individually mean hydrogen, C1-C4 alkyl, fluoro, chloro or bromo, or together with the carbon atom to which they are bound form C3-C6 cycloalkyl group; R6 & R8, independent from each other and individually mean hydrogen, C1-C4 alkyl, fluoro, chloro or bromo, or when R2 & R4 do not form part of a cycloalkyl group R2 & R4 together with the carbon atoms to which they are bound can form C5-C7 cycloalkyl group; and R7 is hydrogen, C1-C4 alkyl, optionally substituted by one or more halo, or C1-C- alkoxy. The invention also relates to their pharmaceutically, veterinary or agriculturally acceptable salts or solvates. 24 claims</p>
申请公布号 BG64127(B1) 申请公布日期 2004.01.30
申请号 BG19990103454 申请日期 1999.06.01
申请人 PFIZER INC. 发明人 BANKS, BERNARD J.
分类号 A01N43/56;A61K31/415;A61K31/4427;A61K31/4439;A61P33/00;C07D231/12;C07D231/14;C07D231/16;C07D231/18;C07D231/38;C07D401/04;(IPC1-7):C07D231/38 主分类号 A01N43/56
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