发明名称 NOVEL FUSED IMIDAZOLE DERIVATIVE
摘要 A compound represented by the general formula (I) [wherein T<1> means an optionally substituted, monocyclic or bicyclic, 4- to 12-membered, heterocyclic group containing one or two nitrogen atoms in the ring; X means optionally substituted C1-6 alkyl, etc.; Z<1> and Z<2> each independently means nitrogen or a group represented by the formula -CR<2>-; and R<1> and R<2> each independently means hydrogen, optionally substituted C1-6 alkyl, optionally substituted C1-6 alkoxy, etc.], a salt of the compound, or a hydrate of either. These are novel compounds having excellent DPPIV inhibitory activity.
申请公布号 WO03104229(A1) 申请公布日期 2003.12.18
申请号 WO2003JP07010 申请日期 2003.06.03
申请人 EISAI CO., LTD.;YOSHIKAWA, SEIJI;EMORI, EITA;MATSUURA, FUMIYOSHI;RICHARD, CLARK;IKUTA, HIRONORI;KIRA, KAZUNOBU;YASUDA, NOBUYUKI;NAGAKURA, TADASHI;YAMAZAKI, KAZUTO 发明人 YOSHIKAWA, SEIJI;EMORI, EITA;MATSUURA, FUMIYOSHI;RICHARD, CLARK;IKUTA, HIRONORI;KIRA, KAZUNOBU;YASUDA, NOBUYUKI;NAGAKURA, TADASHI;YAMAZAKI, KAZUTO
分类号 C07D471/04;A61K31/496;A61K31/5025;A61K31/522;A61K31/5377;A61K31/541;A61P1/00;A61P3/04;A61P3/06;A61P3/10;A61P9/00;A61P15/00;A61P15/08;A61P19/02;A61P19/10;A61P29/00;A61P31/18;A61P35/00;A61P37/00;A61P37/02;A61P37/08;A61P43/00;C07D473/04;C07D473/06;C07D473/18;C07D473/22;C07D473/24;C07D473/30;C07D473/36;C07D473/40;C07D487/04;C07D491/14;(IPC1-7):C07D471/04;C07D498/14;A61K31/502;A61K31/536;A61K31/519 主分类号 C07D471/04
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