发明名称 COMBINATORIAL LIBRARIES OF GEMINALLY SUBSTITUTED AMINES
摘要 The present invention relates to a combinatorial library that comprises amines of the general formula (I) in which R<1>, R<2> and R<3> may be the same or different and represent hydrogen or a substituted or non-substituted alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkinyl or aryl group, -Si(R)3, -Sn(R)3, -SR, -OR or -NRR'. The radicals R<1> and R<2> or R<2> and R<3> can also form together a cycloalkyl ring which may also contain, together with N, at least one other heteroatom, preferably N, O or S. The radicals R<4> and R<5> may be the same or different and represent a substituted or non-substituted alkyl, cycloalkyl, alkenyl, cycloalkenyl, alkinyl or aryl group, -Si(R)3, -Sn(R)3, -SR, -OR or -NRR'. The radicals R<4> and R<5> can also form together a cycloalkyl ring which may also contain, together with N, at least one other heteroatom, preferably N, O or S. In the above-mentioned definition of radicals R<1> to R<5>, R and R' may be the same or different and represent a substituted or non-substituted alkyl radical or a substituted or non-substituted aryl radical.
申请公布号 WO9965855(A3) 申请公布日期 2003.12.11
申请号 WO1999EP04255 申请日期 1999.06.18
申请人 MERCK PATENT GMBH;BUCHHOLZ, HERWIG;WELZ-BIERMANN, URS 发明人 BUCHHOLZ, HERWIG;WELZ-BIERMANN, URS
分类号 C07D295/02;B01J31/02;B01J31/12;C07B61/00;C07C209/66;C07C209/68;C07C209/78;C07C211/05;C07C211/06;C07C211/08;C07C211/16;C07C211/17;C07C211/21;C07C211/22;C07C211/27;C07C211/35;C07C211/48;C07D295/023;C07D295/03;C07D295/06;C07F7/10;C40B40/04;C40B50/00 主分类号 C07D295/02
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