发明名称 PROCESS FOR THE PREPARATION OF OMEPRAZOLE PROCESS FOR THE PREPARATION OF OMEPRAZOLE
摘要 Omeprazole, an anti-ulcer agent having the formula Ia: (see formula Ia) is prepared by treating a mixture of pyrmetazole, having the formula IIa: (see formula IIa) in a solvent with magnesium monoperoxyphthalate, in an amount sufficient to convert pyrmetazole to omeprazole.
申请公布号 CA2078517(C) 申请公布日期 2003.11.04
申请号 CA19922078517 申请日期 1992.09.17
申请人 发明人 HOERRNER, ROBERT SCOTT;FRIEDMAN, JOEL JAY;AMATO, JOSEPH SEBASTIAN;LIU, THOMAS MENG-HAN;SHINKAI, ICHIRO;WEINSTOCK, LEONARD MAURICE
分类号 A61K31/415;A61P1/04;C07D401/12;C07D471/04;(IPC1-7):C07D401/12;C07D405/14;C07D413/14;C07D417/14 主分类号 A61K31/415
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