发明名称 |
PROCESS FOR THE PREPARATION OF OMEPRAZOLE PROCESS FOR THE PREPARATION OF OMEPRAZOLE |
摘要 |
Omeprazole, an anti-ulcer agent having the formula Ia: (see formula Ia) is prepared by treating a mixture of pyrmetazole, having the formula IIa: (see formula IIa) in a solvent with magnesium monoperoxyphthalate, in an amount sufficient to convert pyrmetazole to omeprazole.
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申请公布号 |
CA2078517(C) |
申请公布日期 |
2003.11.04 |
申请号 |
CA19922078517 |
申请日期 |
1992.09.17 |
申请人 |
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发明人 |
HOERRNER, ROBERT SCOTT;FRIEDMAN, JOEL JAY;AMATO, JOSEPH SEBASTIAN;LIU, THOMAS MENG-HAN;SHINKAI, ICHIRO;WEINSTOCK, LEONARD MAURICE |
分类号 |
A61K31/415;A61P1/04;C07D401/12;C07D471/04;(IPC1-7):C07D401/12;C07D405/14;C07D413/14;C07D417/14 |
主分类号 |
A61K31/415 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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