| 发明名称 |
Isothiazole derivatives useful as anticancer agents |
| 摘要 |
The present invention relates to compounds of the formula 1 and to pharmaceutically acceptable salts, prodrugs and solvates thereof, wherein X1, R1, R2 and R3 are as defined herein. The invention also relates to pharmaceutical compositions containing the above compounds and to methods treating hyperproliferative disorders in mammals by administering the above compounds.
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| 申请公布号 |
US2003149048(A1) |
申请公布日期 |
2003.08.07 |
| 申请号 |
US20030357093 |
申请日期 |
2003.02.03 |
| 申请人 |
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发明人 |
LARSON ERIC R.;NOE MARK C.;GANT THOMAS G. |
| 分类号 |
C07D275/02;A61K31/425;A61K31/427;A61K31/454;A61K31/496;A61K45/00;A61P13/08;A61P17/00;A61P35/00;A61P43/00;C07C33/46;C07C323/60;C07C327/58;C07D209/00;C07D275/03;C07D417/12;C07D487/08;C07D521/00;(IPC1-7):A61K31/496;C07D417/02 |
主分类号 |
C07D275/02 |
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