发明名称 5'-ACYLAMINO-1,1'-BIPHENYL-4-CARBOXAMIDE DERIVATIVES AND THEIR USE AS P38 KINASE INHIBITORS
摘要 Compounds of formula (I): wherein R<sp>3</sp> is the group −NH−CO−R<sp>6</sp>; or pharmaceutically acceptable salts or solvates thereof, and their use as pharmaceuticals, particularly as p38 kinase inhibitors.
申请公布号 WO03032971(A1) 申请公布日期 2003.04.24
申请号 WO2002EP11576 申请日期 2002.10.16
申请人 GLAXO GROUP LIMITED;ANGELL, RICHARD, MARTYN;ASTON, NICOLA, MARY;BAMBOROUGH, PAUL;BAMFORD, MARK, JAMES;COCKERILL, GEORGE, STUART;FLACK, STEPHEN, SEAN;LAINE, DRAMANE, IBRAHIM;MERRICK, SUZANNE, JOY;SMITH, KATHRYN, JANE;WALKER, ANN, LOUISE 发明人 ANGELL, RICHARD, MARTYN;ASTON, NICOLA, MARY;BAMBOROUGH, PAUL;BAMFORD, MARK, JAMES;COCKERILL, GEORGE, STUART;FLACK, STEPHEN, SEAN;LAINE, DRAMANE, IBRAHIM;MERRICK, SUZANNE, JOY;SMITH, KATHRYN, JANE;WALKER, ANN, LOUISE
分类号 A61K31/167;A61K31/341;A61K31/351;A61K31/381;A61K31/40;A61K31/402;A61K31/4155;A61K31/42;A61K31/4406;A61K31/4409;A61K31/4436;A61K31/4439;A61K31/4545;A61K31/4709;A61K31/496;A61K31/505;A61K31/5377;A61P1/04;A61P3/10;A61P7/02;A61P9/00;A61P9/04;A61P9/10;A61P11/00;A61P11/06;A61P13/12;A61P17/04;A61P17/06;A61P19/02;A61P19/06;A61P19/08;A61P19/10;A61P21/00;A61P21/04;A61P25/00;A61P25/06;A61P25/08;A61P25/14;A61P25/16;A61P25/28;A61P27/02;A61P27/16;A61P29/00;A61P31/04;A61P31/06;A61P31/18;A61P33/00;A61P33/06;A61P35/00;A61P37/06;A61P37/08;A61P43/00;C07C231/02;C07C231/14;C07C237/42;C07D207/06;C07D207/12;C07D207/26;C07D207/27;C07D207/32;C07D207/327;C07D213/81;C07D213/82;C07D215/50;C07D239/28;C07D239/42;C07D241/04;C07D241/24;C07D241/26;C07D261/18;C07D277/56;C07D307/16;C07D307/24;C07D307/54;C07D307/68;C07D309/08;C07D333/38;C07D401/04;C07D403/04;C07D405/04;C07D409/04;C07D417/04;(IPC1-7):A61K31/166 主分类号 A61K31/167
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