发明名称 |
Apicidin-derived cyclic tetrapeptides |
摘要 |
Cyclic tetrapeptide compounds derived from apicidin therapeutically inhibit histone deacetylase activity, are represented by Formula I: and are useful in the treatment of protozoal infections.
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申请公布号 |
US2003078369(A1) |
申请公布日期 |
2003.04.24 |
申请号 |
US20020066451 |
申请日期 |
2002.01.31 |
申请人 |
MEINKE PETER T.;SCHMATZ DENNIS;MYERS ROBERT W.;RATTRAY SANDRA J.;COLLETTI STEVEN L.;WYVRATT MATTHEW J.;FISHER MICHAEL H.;GURNETT ANNE M. |
发明人 |
MEINKE PETER T.;SCHMATZ DENNIS;MYERS ROBERT W.;RATTRAY SANDRA J.;COLLETTI STEVEN L.;WYVRATT MATTHEW J.;FISHER MICHAEL H.;GURNETT ANNE M. |
分类号 |
A61K38/00;C07K5/12;(IPC1-7):C07K7/54;C07D245/00 |
主分类号 |
A61K38/00 |
代理机构 |
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代理人 |
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