PROCESS FOR PREPARING CHIRAL DIOL SULFONES AND DIHYDROXY ACID HMG COA REDUCTASE INHIBITORS
摘要
A process is provided for preparing chiral diol sulfones of the structure (I) where R3 is preferably (II) or (III) where R4a is preferably aryl such as phenyl, and R1a is preferably alkyl such as t-butyl, which are intermediates used in preparing HMG CoA reductase inhibitors.
申请公布号
WO02098854(A3)
申请公布日期
2003.03.27
申请号
WO2002US17269
申请日期
2002.05.30
申请人
BRISTOL-MYERS SQUIBB COMPANY;BRODFUEHRER, PAUL, R.;SATTELBERG, THOMAS, R., SR.;KANT, JOYDEEP;QIAN, XINHUA
发明人
BRODFUEHRER, PAUL, R.;SATTELBERG, THOMAS, R., SR.;KANT, JOYDEEP;QIAN, XINHUA