发明名称 |
DERIVATIVES OF 4,5-DIARYL-3(2)-FURANONE AS INHIBITORS OF CYKOXYGENEASE-2 |
摘要 |
The present invention provides a novel class of 4,5-diaryl-3(2H)-furanone derivatives, which inhibit strongly and selectively COX-2 over COX-1. They are useful to treat inflammation, inflammation-associated disorders, and COX-2 mediated diseases. |
申请公布号 |
PL351125(A1) |
申请公布日期 |
2003.03.24 |
申请号 |
PL20000351125 |
申请日期 |
2000.04.12 |
申请人 |
PACIFIC CORP. |
发明人 |
SHIN SONG SEOK;NOH MIN-SOO;BYUN YOUNG JOO;CHOI JIN KYU;KIM JIN KWAN;LIM KYUNG MIN;KIM JI YOUNG;CHOI YOUNG HOON;HA JUN-YONG;LEE KI-WHA;MOH JOO HYUN;JEONG YEON SU;CHUNG SHIN;JOO YUNG HYUP;LEE CHANG HOON;KANG SEON HWA;PARK YOUNG-HO;YI JUNG BUM |
分类号 |
A61K31/341;A61K31/343;A61K31/35;A61K31/36;A61K31/381;A61K31/4155;A61K31/443;A61P9/10;A61P25/28;A61P27/02;A61P29/00;A61P35/00;A61P43/00;C07D307/32;C07D307/58;C07D307/64;C07D307/94;C07D405/04;C07D407/04;C07D407/10;C07D409/04;C07D493/10 |
主分类号 |
A61K31/341 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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