发明名称 |
DERIVATIVES OF ARYL(OR HETEROARYL) AZOLYLCARBINOLS FOR THE TREATEMENT OFURINARY INCONTINENCE |
摘要 |
The invention relates to aryl (or heteroaryl) azolylcarbynol derivatives having general formula (I), wherein: Ar represents an optionally substituted phenyl radical or thienyl radical; R1191 represents a hydrogen atom or a low er alkyl group; R2191 represents a dialkylaminoalkyl or azaheterocycloalkyl radical; and Het represents a non-substituted azole or an azole optionally substituted by one or two substituents. The invention also relates to the physiologically-acceptable salts of said derivatives. The inventive derivatives can be used as medicaments in human and/or veterinary therapy fo r the treatment of urinary incontinence in mammals, including humans.
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申请公布号 |
CA2452646(A1) |
申请公布日期 |
2003.01.16 |
申请号 |
CA20022452646 |
申请日期 |
2002.07.01 |
申请人 |
LABORATORIOS DEL DR. ESTEVE, S.A. |
发明人 |
MERCE-VIDAL, RAMON;ANDALUZ-MATARO, BLAS;FRIGOLA-CONSTANSA, JORDI |
分类号 |
C07D231/12;A61K31/40;A61K31/415;A61K31/4155;A61K31/4164;A61K31/4196;A61P7/12;A61P13/10;C07D409/06;(IPC1-7):A61K31/415 |
主分类号 |
C07D231/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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