发明名称 CRYSTALLINE SALTS OF 2-(4-{2-[2-HYDROXY-3-(2-THIOPHEN-2-YL-PHENOXY)-PROPYLAMINO]-2-METHYL-PROPYL}-PHENOXY)-NICOTINONITRILE
摘要 The present invention relates to crystalline salts of 2-(4-{2-[2-hydroxy-3-(2-thiophen-2-yl-phenoxy)-propylamino]-2-methyl-propyl}-phenoxy)-nicotinonitrile. The salts of the present invention, being beta 3 adrenergic receptor agonists, are capable of increasing lipolysis and energy expenditure in cells and, therefore, are useful, e.g., for treating type 2 diabetes and/or obesity.
申请公布号 WO02094820(A1) 申请公布日期 2002.11.28
申请号 WO2002US11896 申请日期 2002.05.20
申请人 ELI LILLY AND COMPANY;BUSH, JULIE, KAY;REMICK, DAVID, MICHAEL 发明人 BUSH, JULIE, KAY;REMICK, DAVID, MICHAEL
分类号 C07D207/32;C07D207/333;C07D213/30;C07D213/82;C07D213/84;C07D261/08;C07D277/24;C07D333/16;C07D401/12;C07D405/12;C07D409/12;C07D413/12;C07D417/12;(IPC1-7):C07D409/12;A61K31/44 主分类号 C07D207/32
代理机构 代理人
主权项
地址