发明名称 |
Process for the preparation of chemical compounds |
摘要 |
An improved and efficient synthesis for the preparation of 2-amino-6-[(4-aminopiperidin-1-yl]methyl]pyridine, an intermediate compound in the preparation of muscarinic M3 receptor antagonists, includes as a final step the removal of trimethylacetyl and an amino protecting group from 2-trimethylacetyl-amino-6-[(4-protected aminopiperidin-1-yl)methyl]pyridine.
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申请公布号 |
US6469172(B2) |
申请公布日期 |
2002.10.22 |
申请号 |
US20010799440 |
申请日期 |
2001.03.05 |
申请人 |
MERCK & CO., INC. |
发明人 |
MALIGRES PETER E.;LEE JAEMOON |
分类号 |
C07D401/06;(IPC1-7):C07D401/06 |
主分类号 |
C07D401/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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