发明名称 PROCESS FOR PREPARING 3-ARYL-BENZO[B]THIOPHENES
摘要 The present invention relates to a process for preparing a compound of formula (I): which includes cyclodehydrating a compound of formula (II): in the presence of an acid activated clay or acid activated zeolite catalyst and in the presence of a suitable solvent.
申请公布号 WO0242289(A3) 申请公布日期 2002.09.06
申请号 WO2001US42940 申请日期 2001.11.14
申请人 ELI LILLY AND COMPANY;LUKE, WAYNE, DOUGLAS;SANDERSON, HEIDI, ANN;ZHENG, HUA 发明人 LUKE, WAYNE, DOUGLAS;SANDERSON, HEIDI, ANN;ZHENG, HUA
分类号 C07D333/52;C07D333/56;C07D333/64;C07D409/00 主分类号 C07D333/52
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