发明名称 |
FARNESYL TRANSFERASE INHIBITING BENZOHETEROCYCLIC DERIVATIVES |
摘要 |
This invention comprises the novel compounds of formula (I) wherein r, s, t, X, Z, R<1>, R<2>, R<3>, R<4>, R<5>, R<6> and R<7> have defined meanings, having farnesyl transferase inhibiting activity; their preparation, compositions containing them and their use as a medicine.
|
申请公布号 |
WO0242296(A1) |
申请公布日期 |
2002.05.30 |
申请号 |
WO2001EP13317 |
申请日期 |
2001.11.15 |
申请人 |
JANSSEN PHARMACEUTICA N.V.;ANGIBAUD, PATRICK, RENE;VENET, MARC, GASTON;PONCELET, VIRGINIE, SOPHIE |
发明人 |
ANGIBAUD, PATRICK, RENE;VENET, MARC, GASTON;PONCELET, VIRGINIE, SOPHIE |
分类号 |
A61K31/395;A61K31/5513;A61K31/553;A61K31/554;A61P1/04;A61P3/04;A61P3/10;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P11/16;A61P15/00;A61P17/00;A61P17/04;A61P17/06;A61P17/10;A61P17/14;A61P19/02;A61P19/06;A61P19/08;A61P25/00;A61P27/02;A61P29/00;A61P31/12;A61P31/18;A61P33/06;A61P35/00;A61P37/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D403/06;C07D413/06;C07D417/06;C07D498/04;(IPC1-7):C07D413/06;A61K31/551 |
主分类号 |
A61K31/395 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|