发明名称 |
SULFONYL AMINO DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME |
摘要 |
<p>The invention relates to sulfonyl amine derivatives of formula IA wherein R<SUP>5A</SUP>, X<SUP>1</SUP>, X<SUP>2</SUP>, R<SUP>9 </SUP>and R<SUP>10 </SUP>are as defined herein, which derivatives are useful as bradykinin B<SUB>1 </SUB>receptor antagonists.</p> |
申请公布号 |
SK17492001(A3) |
申请公布日期 |
2002.04.04 |
申请号 |
SK20010001749 |
申请日期 |
2000.06.02 |
申请人 |
NOVARTIS AG |
发明人 |
BRAIN CHRISTOPHER THOMAS;CANTRELL WILLIAM;CULSHAW ANDREW JAMES;DZIADULEWICZ EDWARD KAROL;HART TERANCE WILLIAM;RITCHIE TIMOTHY JOHN;WAYKOLE LILADHAR |
分类号 |
C07D295/18;A61K31/4406;A61K31/4409;A61K31/496;A61K31/5377;A61K31/541;A61K31/63;A61P1/04;A61P1/18;A61P7/10;A61P9/02;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/10;A61P15/00;A61P15/06;A61P17/00;A61P17/02;A61P17/04;A61P17/06;A61P19/02;A61P19/04;A61P19/06;A61P21/00;A61P21/02;A61P25/00;A61P25/02;A61P25/04;A61P25/06;A61P25/08;A61P27/02;A61P29/00;A61P31/04;A61P35/00;A61P37/08;A61P41/00;A61P43/00;C07C311/44;C07D211/34;C07D211/62;C07D211/82;C07D213/38;C07D261/08;C07D277/28;C07D295/192;C07D295/26;C07D333/20;C07D401/12;(IPC1-7):C07C311/44 |
主分类号 |
C07D295/18 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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