发明名称 BICYCLYL OR HETEROBICYCLYLMETHANESULFONYLAMINO-SUBSTITUTED N-HYDROXYFORMAMIDES
摘要 Compounds of formula (I): R is hydrogen, alkyl, alkenyl, alkynyl, aryl, heteroaryl or heterocyclyl; and R1 is bicyclyl or heterobicyclyl, are useful in the treatment and prophylaxis of conditions mediated by s-CD23.
申请公布号 CA2410294(A1) 申请公布日期 2001.11.29
申请号 CA20012410294 申请日期 2001.05.21
申请人 SMITHKLINE BEECHAM P.L.C. 发明人 BRUTON, GORDON;ORLEK, BARRY SIDNEY;BEST, DESMOND JOHN;WALKER, GRAHAM;RANA, KISHORE
分类号 C07D333/38;A61K31/16;A61K31/343;A61K31/381;A61K31/4155;A61K31/422;A61K31/428;A61K31/437;A61K31/47;A61K31/4709;A61K31/538;A61P7/02;A61P7/04;A61P9/00;A61P11/06;A61P17/00;A61P25/28;A61P27/14;A61P27/16;A61P29/00;A61P31/00;A61P37/00;A61P37/06;A61P37/08;A61P43/00;C07C315/02;C07C315/04;C07C317/28;C07C323/29;C07D215/12;C07D215/14;C07D277/62;C07D307/79;C07D307/81;C07D333/54;C07D333/58;C07D333/60;C07D333/62;C07D405/12;C07D409/12;C07D413/12;C07D495/04;(IPC1-7):C07D333/60 主分类号 C07D333/38
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