发明名称 MACROCYCLIC NS3-SERINE PROTEASE INHIBITORS OF HEPATITIS C VIRUS COMPRISING N-CYCLIC P2 MOIETIES
摘要 The present invention discloses novel macrocyclic compounds which have HCV protease inhibitory activity as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising such macrocycles as well as methods of using them to treat disorders associated with the HCV protease.
申请公布号 WO0177113(A2) 申请公布日期 2001.10.18
申请号 WO2001US10869 申请日期 2001.04.03
申请人 SCHERING CORPORATION 发明人 CHEN, KEVIN, X.;ARASAPPAN, ASHOK;VENKATRAMAN, SRIKANTH;PAREKH, TEJAL, N.;GU, HAINING;NJOROGE, F., GEORGE;GIRIJAVALLABHAN, VIYYOOR, M.;GANGULY, ASHIT;SAKSENA, ANIL;JAO, EDWIN;YAO, NANHUA, H.;PRONGAY, ANDREW, J.;MADISON, VINCENT, S.;VIBULBHAN, BANCHA
分类号 C12N9/99;A61K31/7052;A61K38/00;A61K38/21;A61K38/55;A61K45/00;A61P31/12;A61P31/14;A61P43/00;C07K1/02;C07K5/023;C07K5/08;C07K5/083;C07K5/12;C07K7/02;(IPC1-7):C07D498/00 主分类号 C12N9/99
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