SOLID-SUPPORTED PROCESS FOR MAKING N-SUBSTITUTED PEPTIDE MIMETIC COMPOUNDS
摘要
The subject invention involves processes for making N-substituted peptide mimetic compounds comprising a Petasis reaction scheme using reactants comprising an activated carbonyl compound, an amine compound, and a boronic acid compound, and libraries of such compounds.
申请公布号
WO0155091(A1)
申请公布日期
2001.08.02
申请号
WO2001US02467
申请日期
2001.01.25
申请人
THE PROCTER & GAMBLE COMPANY;KLOPFENSTEIN, SEAN, REES;GOLEBIOWSKI, ADAM;LI, MIN
发明人
KLOPFENSTEIN, SEAN, REES;GOLEBIOWSKI, ADAM;LI, MIN