发明名称 PHOSPHONIC ACID BIARYL DERIVATIVES AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE 1B (PTP-1B)
摘要 The invention encompasses the novel class of compounds represented by formula (I), which are inhibitors of the PTP-1B enzyme. The invention also encompasses pharmaceutical compositions and methods of treating or preventing PTP-1B mediated diseases, including diabetes, obesity, and diabetes-related conditions.
申请公布号 WO0146203(A1) 申请公布日期 2001.06.28
申请号 WO2000CA01547 申请日期 2000.12.21
申请人 MERCK FROSST CANADA & CO.;LAU, CHEUK, KUN;BAYLY, CHRISTOPHER;GAUTHIER, JACQUES, YVES;LEBLANC, YVES;LI, CHUN, SING;ROY, PATRICK;THERIEN, MICHEL;WANG, ZHAOYIN 发明人 LAU, CHEUK, KUN;BAYLY, CHRISTOPHER;GAUTHIER, JACQUES, YVES;LEBLANC, YVES;LI, CHUN, SING;ROY, PATRICK;THERIEN, MICHEL;WANG, ZHAOYIN
分类号 A61K45/00;A61K31/675;A61P1/04;A61P1/18;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P25/28;A61P35/00;A61P43/00;C07F9/60;C07F9/6518;C07F9/6558;C07F9/6561;(IPC1-7):C07F9/38;A61K31/66;C07F9/553;C07F9/653;C07F9/651;C07F9/652;C07F9/654;C07F9/650 主分类号 A61K45/00
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