发明名称 |
Inhibitors of neuraminidases |
摘要 |
Disclosed are compounds of the formula:which are useful for inhibiting neuraminidases from disease-causing microorganisms, especially, influenza neuraminidase. Also disclosed are compositions and methods for preventing and treating diseases caused by microorganisms having a neuraminidase, processes for preparing the compounds and synthetic intermediates used in these processes. |
申请公布号 |
AU1076001(A) |
申请公布日期 |
2001.04.30 |
申请号 |
AU20010010760 |
申请日期 |
2000.10.10 |
申请人 |
ABBOTT LABORATORIES |
发明人 |
CLARENCE J. MARING;VINCENT L. GIRANDA;DALE J. KEMPF;VINCENT S. STOLL;MINGHUA SUN;CHEN ZHAO;YU GUI GU;STEPHEN HANESSIAN;GARY T WANG;ALLAN C. KRUEGER;HUI-JU CHEN;YUANWEI CHEN;DAVID A. DEGOEY;WILLIAM J. FLOSI;DAVID J. GRAMPOVNIK;WARREN M. KATI;APRIL L. KENNEDY;LARRY L. KLEIN;ZHEN LIN;DAROLD L. MADIGAN;KEITH F. MCDANIEL;STEVEN W. MUCHMORE;HING L. SHAM;KENT D. STEWART;NOAH P. TU;FRANK L. WAGENAAR;SHELDON WANG;PAUL E. WIEDEMAN;YIBO XU;MING C. YEUNG;MALKEN BAYRAKDARIAN;XUEHONG LUO |
分类号 |
C07D401/12;A61K31/357;A61K31/40;A61K31/401;A61K31/4025;A61K31/405;A61K31/415;A61K31/4155;A61K31/4178;A61K31/42;A61K31/422;A61K31/425;A61K31/427;A61K31/4439;A61K31/5377;A61K31/66;A61K31/662;A61P31/00;A61P31/12;A61P31/16;A61P43/00;C07D;C07D207/00;C07D207/12;C07D207/16;C07D207/26;C07D207/32;C07D207/327;C07D207/38;C07D207/46;C07D303/16;C07D403/04;C07D403/06;C07D405/04;C07D405/06;C07D407/06;C07D407/12;C07D409/06;C07D413/04;C07D413/06;C07D417/04;C07D417/06;C07D521/00;C07F9/40;C07F9/572 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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