发明名称 PROCESS FOR THE PREPARATION OF PYRAZOLO [4,3-D] PYRIMIDIN-7-ONES-3-PYRIDYLSULPHONYL COMPOUNDS AND INTERMEDIATES THEREOF
摘要 A process is provided for the preparation of compounds of formula (I) herein comprising reacting a compound of formula (II), (III) or (IV) in the presence of <->OR and a hydroxide trapping agent or in the case of compounds of formula (IV) reacting in the presence of an auxiliary base and a hydroxide trapping agent (i.e. <->OR is substituted by the auxiliary base), wherein X is a leaving group and R<1> to R<4> are as defined above.
申请公布号 EA200000924(A2) 申请公布日期 2001.04.23
申请号 EA20000000924 申请日期 2000.10.10
申请人 发明人
分类号 A61K;C07D;C07D213/83;C07D401/12;C07D401/14;C07D487/04 主分类号 A61K
代理机构 代理人
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