发明名称 |
Benzopyran-containing compounds and method for their use |
摘要 |
Certain benzopyran antiestrogens are disclosed for treating estrogen sensitive diseases such as breast cancer. Prodrug forms provide ease of manufacturing, good shelf life, and bioavailability, and preferred stereoisomers are shown to be more effective than racemic mixtures.
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申请公布号 |
US6060503(A) |
申请公布日期 |
2000.05.09 |
申请号 |
US19950388207 |
申请日期 |
1995.02.21 |
申请人 |
ENDORECHERCHE, INC. |
发明人 |
LABRIE, FERNAND;MERAND, YVES;GAUTHIER, SYLVAIN |
分类号 |
C07D405/12;A61K31/10;A61K31/135;A61K31/138;A61K31/165;A61K31/35;A61K31/352;A61K31/353;A61K31/38;A61K31/382;A61K31/40;A61K31/4025;A61K31/445;A61K31/4453;A61K31/453;A61K31/4535;A61K31/47;A61K31/4709;A61K31/472;A61K31/4725;A61P35/00;C07C215/64;C07C217/18;C07C235/34;C07C317/18;C07D215/14;C07D217/16;C07D295/092;C07D295/096;C07D295/185;C07D311/60;C07D335/06;C07J1/00;C07J17/00;C07J21/00;C07J41/00;C07J51/00;C07J53/00;C07J71/00;(IPC1-7):A61K31/40;A61K31/44 |
主分类号 |
C07D405/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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