发明名称 Benzopyran-containing compounds and method for their use
摘要 Certain benzopyran antiestrogens are disclosed for treating estrogen sensitive diseases such as breast cancer. Prodrug forms provide ease of manufacturing, good shelf life, and bioavailability, and preferred stereoisomers are shown to be more effective than racemic mixtures.
申请公布号 US6060503(A) 申请公布日期 2000.05.09
申请号 US19950388207 申请日期 1995.02.21
申请人 ENDORECHERCHE, INC. 发明人 LABRIE, FERNAND;MERAND, YVES;GAUTHIER, SYLVAIN
分类号 C07D405/12;A61K31/10;A61K31/135;A61K31/138;A61K31/165;A61K31/35;A61K31/352;A61K31/353;A61K31/38;A61K31/382;A61K31/40;A61K31/4025;A61K31/445;A61K31/4453;A61K31/453;A61K31/4535;A61K31/47;A61K31/4709;A61K31/472;A61K31/4725;A61P35/00;C07C215/64;C07C217/18;C07C235/34;C07C317/18;C07D215/14;C07D217/16;C07D295/092;C07D295/096;C07D295/185;C07D311/60;C07D335/06;C07J1/00;C07J17/00;C07J21/00;C07J41/00;C07J51/00;C07J53/00;C07J71/00;(IPC1-7):A61K31/40;A61K31/44 主分类号 C07D405/12
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